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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T4983 | Isoetharine mesylate salt | Isoetarine mesilate | Others , Adrenergic Receptor |
Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression. | |||
T24579 | Oxyfedrine L-form HCl | Modacor,Oxyfedrine L-form hydrochloride,D563,Ildamen,D 563,D-563 | Adrenergic Receptor |
Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent. | |||
T30504 | BMS-196085 | SCHEMBL7042488,BMS196085,CHEMBL322862,FM0D5L3W03 | |
BMS-196085 is an effective and selective human β( 3) All agonists of adrenergic receptors, in β( 1) Partial agonist activity was 45%. | |||
T68114 | Nardeterol | ||
Nardeterol is a high-affinity, partial agonist for beta adrenergic receptors. | |||
T14498 | Barbadin | Arrestin | |
Barbadin is a novel and specific inhibitor of β-arrestin/β2-adaptin interaction with an IC50 value of 19.1 μM for β-arestin1 and 15.6 μM for β-arestin2. Barbadin potentiates the long term effects of lorcaserin on POMC ne... |